Susan Lepri

Indole Based Weapons to Fight Antibiotic Resistance: A Structure–Activity Relationship Study

Susan Lepri, Federica Buonerba, Laura Goracci et al. · Journal of Medicinal Chemistry · 2016 · 76 citations · Full text

Pharmaceutical Science, Antibiotic Resistance, Pharmaceutical Chemistry +16

Discovery of a Chemical Probe Bisamide (CCT251236): An Orally Bioavailable Efficacious Pirin Ligand from a Heat Shock Transcription Factor 1 (HSF1) Phenotypic Screen

Matthew D. Cheeseman, N. Chessum, Carl S. Rye et al. · Journal of Medicinal Chemistry · 2016 · 67 citations · Full text

Medicinal Chemistry, Phenotypic Screens, Drug Target +13

Rotational barriers of biphenyls having heavy heteroatoms as ortho-substituents: experimental and theoretical determination of steric effects

Lodovico Lunazzi, Michele Mancinelli, Andrea Mazzanti et al. · Organic & Biomolecular Chemistry · 2011 · 65 citations · Full text

Engineering, Organic Chemistry, Computational Chemistry +16

Optimization of Small-Molecule Inhibitors of Influenza Virus Polymerase: From Thiophene-3-Carboxamide to Polyamido Scaffolds

Susan Lepri, Giulio Nannetti, Giulia Muratore et al. · Journal of Medicinal Chemistry · 2014 · 62 citations

Structure–metabolism relationships in <i>human-</i> AOX: Chemical insights from a large database of aza-aromatic and amide compounds

Susan Lepri, Martina Ceccarelli, Nicolò Milani et al. · Proceedings of the National Academy of Sciences · 2017 · 55 citations · Full text