Roberto Perrone

Cyclohexylpiperazine derivative PB28, a σ2 agonist and σ1 antagonist receptor, inhibits cell growth, modulates P-glycoprotein, and synergizes with anthracyclines in breast cancer

Amalia Azzariti, Nicola Antonio Colabufo, Francesco Berardi et al. · Molecular Cancer Therapeutics · 2006 · 113 citations · Full text

Breast Oncology, Low Sigma, Chemoprevention Strategy +19

Antiproliferative and cytotoxic effects of some ?2 agonists and ?1 antagonists in tumour cell lines

NicolaAntonio Colabufo, Francesco Berardi, Marialessandra Contino et al. · Naunyn-Schmiedeberg s Archives of Pharmacology · 2004 · 109 citations

Cytotoxic Effects, Tumour Cell Lines, Chemoprevention Strategy +10

High Affinity and Selectivity on 5-HT1A Receptor of 1-Aryl-4-[(1-tetralin)alkyl]piperazines. 2

Roberto Perrone, Francesco Berardi, Nicola Antonio Colabufo et al. · Journal of Medicinal Chemistry · 1995 · 91 citations · Full text

Small P-gp modulating molecules: SAR studies on tetrahydroisoquinoline derivatives

Nicola Antonio Colabufo, Francesco Berardi, Mariangela Cantore et al. · Bioorganic & Medicinal Chemistry · 2007 · 80 citations · Full text

Medicinal Chemistry, Natural Sciences, Organic Chemistry +4

LP-211 is a brain penetrant selective agonist for the serotonin 5-HT7 receptor

Peter B. Hedlund, Marcello Leopoldo, Silvio Caccia et al. · Neuroscience Letters · 2010 · 77 citations

Functional Selectivity, Medicine, Serotonin 5-Ht7 Receptor +7