Timothy D. Gross

(2,4,6-Triisopropylphenyl)selenium Bromide (TIPPSe-Br). An in Situ-Generated Reagent for Effecting Highly Selective Ring Closures of Homoallylic Alcohols to Substituted Tetrahydrofurans

Bruce H. Lipshutz, Timothy D. Gross · The Journal of Organic Chemistry · 1995 · 54 citations

Situ-generated Reagent, Derivative (Chemistry), Engineering +11

3-[(2<i>R</i>)-Amino-2-phenylethyl]-1-(2,6-difluorobenzyl)-5-(2-fluoro-3-methoxyphenyl)- 6-methylpyrimidin-2,4-dione (NBI 42902) as a Potent and Orally Active Antagonist of the Human Gonadotropin-Releasing Hormone Receptor. Design, Synthesis, and in Vitro and in Vivo Characterization

Fábio C. Tucci, Yunfei Zhu, R. Scott Struthers et al. · Journal of Medicinal Chemistry · 2005 · 53 citations · Full text

Pharmaceutical Science, Substituted Uracils, Peptide Science +20

Synthesis and Structure−Activity Relationships of 1-Arylmethyl-5-aryl-6-methyluracils as Potent Gonadotropin-Releasing Hormone Receptor Antagonists

Zhiqiang Guo, Yunfei Zhu, Timothy D. Gross et al. · Journal of Medicinal Chemistry · 2004 · 44 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Methyl Group +15

Chemical Development of NBI-75043. Use of a Flow Reactor to Circumvent a Batch-Limited Metal−Halogen Exchange Reaction

Timothy D. Gross, Shine Chou, Daniel Bonneville et al. · Organic Process Research & Development · 2008 · 33 citations

Chemical Kinetics, Engineering, Chemical Development +16

A novel synthesis of 7-aryl-8-fluoro-pyrrolo[1,2-a]pyrimid-4-ones as potent, stable GnRH receptor antagonists

Fábio C. Tucci, Yunfei Zhu, Zhiqiang Guo et al. · Bioorganic & Medicinal Chemistry Letters · 2002 · 33 citations · Full text

Biochemistry, Medicine, Pharmacological Agent +4