Timothy D. Gross - Concepedia

Author

Timothy D. Gross

Neurocrine Biosciences (United States)

Also Known As

T. Gross, Timothy D Gross, Timothy D. Gross, Timothy Gross

Publications

653

Citations

H-Index

Concepts

All Affiliations

Neurocrine Biosciences (United States)

About

Timothy D. Gross is an author at Neurocrine Biosciences (United States) specializing in pharmacology, medicine, and drug discovery.

Top Concepts

#	Concept	H-Index	Publications	Citations
1	Medicine	16	19	487
2	Natural Sciences	13	15	383
3	Engineering	5	5	139
4	Language Studies	1	1	18
5	Art History	1	1	18

Timothy D. Gross

Publications

644

Citations

H-Index

Page 1

	Year	Citations
(2,4,6-Triisopropylphenyl)selenium Bromide (TIPPSe-Br). An in Situ-Generated Reagent for Effecting Highly Selective Ring Closures of Homoallylic Alcohols to Substituted Tetrahydrofurans Bruce H. Lipshutz, Timothy D. Gross The Journal of Organic Chemistry Situ-generated ReagentDerivative (Chemistry)EngineeringSelenium BromideOrganic Chemistry	1995	54
3-[(2<i>R</i>)-Amino-2-phenylethyl]-1-(2,6-difluorobenzyl)-5-(2-fluoro-3-methoxyphenyl)- 6-methylpyrimidin-2,4-dione (NBI 42902) as a Potent and Orally Active Antagonist of the Human Gonadotropin-Releasing Hormone Receptor. Design, Synthesis, and in Vitro and in Vivo Characterization Fábio C. Tucci, Yunfei Zhu, R. Scott Struthers, Journal of Medicinal Chemistry Pharmaceutical ScienceSubstituted UracilsPeptide SciencePharmacotherapyNbi 42902	2005	53
Synthesis and Structure−Activity Relationships of 1-Arylmethyl-5-aryl-6-methyluracils as Potent Gonadotropin-Releasing Hormone Receptor Antagonists Zhiqiang Guo, Yunfei Zhu, Timothy D. Gross, Journal of Medicinal Chemistry Molecular PharmacologyMedicinal ChemistryMethyl GroupUracil CompoundsBiochemistry	2004	44
Chemical Development of NBI-75043. Use of a Flow Reactor to Circumvent a Batch-Limited Metal−Halogen Exchange Reaction Timothy D. Gross, Shine Chou, Daniel Bonneville, Organic Process Research & Development Chemical KineticsEngineeringChemical DevelopmentChemistryChemical Engineering	2008	33
A novel synthesis of 7-aryl-8-fluoro-pyrrolo[1,2-a]pyrimid-4-ones as potent, stable GnRH receptor antagonists Fábio C. Tucci, Yunfei Zhu, Zhiqiang Guo, Bioorganic & Medicinal Chemistry Letters BiochemistryMedicinePharmacological AgentNovel SynthesisPharmacology	2002	33
Design and Structure−Activity Relationships of 2-Alkyl-3-aminomethyl-6-(3-methoxyphenyl)-7-methyl-8-(2-fluorobenzyl)imidazolo[1,2-<i>a</i>]pyrimid-5-ones as Potent GnRH Receptor Antagonists Yunfei Zhu, Zhiqiang Guo, Timothy D. Gross, Journal of Medicinal Chemistry Drug TargetPharmacotherapyChemical BiologyPharmaceutical ChemistryMolecular Pharmacology	2003	31
Synthesis and initial structure–Activity relationships of a novel series of imidazolo[1,2-a]pyrimid-5-ones as potent GnRH receptor antagonists Keith Wilcoxen, Yun-Fei Zhu, Patrick J. Connors, Bioorganic & Medicinal Chemistry Letters Initial Structure–activity RelationshipsMedicinal ChemistryNovel SeriesBiochemistryMedicine	2002	31
3-(2-Aminoalkyl)-1-(2,6-difluorobenzyl)-5- (2-fluoro-3-methoxyphenyl)-6-methyl- uracils as Orally Bioavailable Antagonists of the Human Gonadotropin Releasing Hormone Receptor Fábio C. Tucci, Yunfei Zhu, Zhiqiang Guo, Journal of Medicinal Chemistry Pharmaceutical SciencePotent Human GonadotropinPharmacotherapyHormone Receptor AntagonistsPharmaceutical Chemistry	2004	29
An Approach to Early-Phase Salt Selection: Application to NBI-75043 Timothy D. Gross, Kevin M. Schaab, Michael A. Ouellette, Organic Process Research & Development EngineeringCorrosionPhase EquilibriumSoil SalinitySalt Selection	2007	28
Initial Structure–Activity Relationship Studies of a Novel Series of Pyrrolo[1,2-a]pyrimid-7-ones as GnRH Receptor Antagonists Yunfei Zhu, R. Scott Struthers, Patrick J. Connors, Bioorganic & Medicinal Chemistry Letters Novel SeriesBiochemistryMedicineMechanism Of ActionReceptor (Biochemistry)	2002	28

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