Rodrigo J. Carbajo

Development of a Novel B-Cell Lymphoma 6 (BCL6) PROTAC To Provide Insight into Small Molecule Targeting of BCL6

William McCoull, Tony Cheung, Erica Anderson et al. · ACS Chemical Biology · 2018 · 133 citations · Full text

Hematological Malignancy, Lymphoid Neoplasia, B-cell Lymphoma 6 +14

Discovery of AZD9833, a Potent and Orally Bioavailable Selective Estrogen Receptor Degrader and Antagonist

James S. Scott, Amber Balazs, Bernard Barlaam et al. · Journal of Medicinal Chemistry · 2020 · 109 citations · Full text

Polymer Masked−Unmasked Protein Therapy. 1. Bioresponsive Dextrin−Trypsin and −Melanocyte Stimulating Hormone Conjugates Designed for α-Amylase Activation

Ruth Duncan, Helena Rosalind Petra Gilbert, Rodrigo J. Carbajo et al. · Biomacromolecules · 2008 · 93 citations

Synthesis of polysubstituted azepanes by dearomative ring expansion of nitroarenes

Rory C. Mykura, Raquel Sánchez-Bento, Esteban Matador et al. · Nature Chemistry · 2024 · 83 citations · Full text

Organic Chemistry, Synthetic Chemistry, Heterocyclic +1

Structure-Based Design and Pharmacokinetic Optimization of Covalent Allosteric Inhibitors of the Mutant GTPase KRAS^G12C

Jason G. Kettle, Sharan K. Bagal, Sue Bickerton et al. · Journal of Medicinal Chemistry · 2020 · 80 citations · Full text