Joseph DiBrino

Synthesis, in vitro and in vivo activity of novel 9-deoxo-9a-aza-9a-homoerythromycin A derivatives; A new class of macrolide antibiotics, the azalides.

G. Michael Bright, A. Nagel, Jon Bordner et al. · The Journal of Antibiotics · 1988 · 238 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

Discovery of 1-[9-(4-Chlorophenyl)-8-(2-chlorophenyl)-9<i>H</i>-purin-6-yl]-4-ethylaminopiperidine-4-carboxylic Acid Amide Hydrochloride (CP-945,598), a Novel, Potent, and Selective Cannabinoid Type 1 Receptor Antagonist

David A. Griffith, John R. Hadcock, Shawn C. Black et al. · Journal of Medicinal Chemistry · 2008 · 64 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

Pyrazolinone-piperidine dipeptide growth hormone secretagogues (GHSs)

Philip A. Carpino, Bruce A. Lefker, Steven M. Toler et al. · Bioorganic & Medicinal Chemistry · 2003 · 47 citations

Medicine, Endocrinology, Pharmacology +12

New bicyclic cannabinoid receptor-1 (CB1-R) antagonists

Philip A. Carpino, David A. Griffith, Subas M. Sakya et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 42 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +12

Discovery and biological characterization of capromorelin analogues with extended half-lives

Philip A. Carpino, Bruce A. Lefker, Steven M. Toler et al. · Bioorganic & Medicinal Chemistry Letters · 2002 · 29 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +8