Gilles H. Goetz

EPSA: A Novel Supercritical Fluid Chromatography Technique Enabling the Design of Permeable Cyclic Peptides

Gilles H. Goetz, Laurence Philippe, Michael J. Shapiro · ACS Medicinal Chemistry Letters · 2014 · 157 citations · Full text

Pharmacy, Pharmaceutics, Pharmacology +15

Resistance factors to grey mould in grape berries: identification of some phenolics inhibitors of Botrytis cinerea stilbene oxidase

Gilles H. Goetz, Abdellatif Fkyerat, Nadine Métais et al. · Phytochemistry · 1999 · 136 citations

Agriculture, Plant Pathology, Plant Sciences +11

High Throughput Method for the Indirect Detection of Intramolecular Hydrogen Bonding

Gilles H. Goetz, William Farrell, Marina Shalaeva et al. · Journal of Medicinal Chemistry · 2014 · 113 citations · Full text

Pharmacy, Chemistry, Pharmaceutical Analysis +15

Discovery of a Novel Class of Exquisitely Selective Mesenchymal-Epithelial Transition Factor (c-MET) Protein Kinase Inhibitors and Identification of the Clinical Candidate 2-(4-(1-(Quinolin-6-ylmethyl)-1 <i>H</i> -[1,2,3]triazolo[4,5- <i>b</i> ]pyrazin-6-yl)-1 <i>H</i> -pyrazol-1-yl)ethanol (PF-04217903) for the Treatment of Cancer

J. Jean Cui, Michele McTigue, Mitchell D. Nambu et al. · Journal of Medicinal Chemistry · 2012 · 105 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Integrating Intramolecular Hydrogen Bonding (IMHB) Considerations in Drug Discovery Using ΔlogP As a Tool

Marina Shalaeva, Giulia Caron, Yuriy A. Abramov et al. · Journal of Medicinal Chemistry · 2013 · 89 citations · Full text

Pharmacy, Chemistry, Medicinal Chemistry +13