Emily F. Calderwood

Substrate-Based Design of the First Class of Angiotensin-Converting Enzyme-Related Carboxypeptidase (ACE2) Inhibitors

Natalie A. Dales, Alexandra E. Gould, James A. Brown et al. · Journal of the American Chemical Society · 2002 · 187 citations · Full text

Life Sciences, Biochemistry, Pharmacology +13

Design and Optimization of Potent and Orally Bioavailable Tetrahydronaphthalene Raf Inhibitors

Alexandra E. Gould, Ruth Adams, Sharmila Adhikari et al. · Journal of Medicinal Chemistry · 2011 · 33 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

Synthesis and biological evaluation of imidazole-based small molecule antagonists of the melanocortin 4 receptor (MC4-R)

Thomas H. Marsilje, Jonathan B Roses, Emily F. Calderwood et al. · Bioorganic & Medicinal Chemistry Letters · 2004 · 33 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

Discovery and optimization of pyrazolopyrimidine sulfamates as ATG7 inhibitors

Shih‐Chung Huang, Sharmila Adhikari, James E. Brownell et al. · Bioorganic & Medicinal Chemistry · 2020 · 31 citations · Full text

Life Sciences, Oncology, Pharmacology +16

Optimization of tetrahydronaphthalene inhibitors of Raf with selectivity over hERG

Shih‐Chung Huang, Sharmila Adhikari, Roushan Afroze et al. · Bioorganic & Medicinal Chemistry Letters · 2016 · 10 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +11