Vincenzo Bernardo

Discovery of the first small molecule inhibitor of human DDX3 specifically designed to target the RNA binding site: Towards the next generation HIV-1 inhibitors

Marco Radi, Federico Falchi, Anna Garbelli et al. · Bioorganic & Medicinal Chemistry Letters · 2012 · 87 citations · Full text

Life Sciences, Medicinal Chemistry, Molecular Biology +17

Design, Synthesis, Biological Activity, and ADME Properties of Pyrazolo[3,4-<i>d</i>]pyrimidines Active in Hypoxic Human Leukemia Cells: A Lead Optimization Study

Marco Radi, Elena Dreassi, Chiara Brullo et al. · Journal of Medicinal Chemistry · 2011 · 82 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Microwave-assisted organocatalytic multicomponent Knoevenagel/hetero Diels–Alder reaction for the synthesis of 2,3-dihydropyran[2,3-c]pyrazoles

Marco Radi, Vincenzo Bernardo, Beatrice Bechi et al. · Tetrahedron Letters · 2009 · 80 citations

Natural Sciences, Chemistry, Medicinal Chemistry +10

Design and Synthesis of Thiadiazoles and Thiazoles Targeting the Bcr‐Abl T315I Mutant: from Docking False Positives to ATP‐Noncompetitive Inhibitors

Marco Radi, Emmanuele Crespan, Federico Falchi et al. · ChemMedChem · 2010 · 21 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17