Alison J. Capolino

Trifluoromethyl group as a pharmacophore: Effect of replacing a CF3 group on binding and agonist activity of a glucocorticoid receptor ligand

Raj Betageri, Yan Zhang, Renée Zindell et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 106 citations · Full text

Medicinal Chemistry, Biochemistry, Medicine +7

Structure−Activity Relationships of the p38α MAP Kinase Inhibitor 1-(5-<i>tert</i>-Butyl-2-<i>p</i>-tolyl-2<i>H</i>-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)naph- thalen-1-yl]urea (BIRB 796)

John R. Regan, Alison J. Capolino, Pier F. Cirillo et al. · Journal of Medicinal Chemistry · 2003 · 105 citations · Full text

Drug Target, Birb 796, Chemical Biology +18

Discovery and SAR study of novel dihydroquinoline-containing glucocorticoid receptor agonists

Hidenori Takahashi, Younes Bekkali, Alison J. Capolino et al. · Bioorganic & Medicinal Chemistry Letters · 2007 · 48 citations · Full text

Biochemistry, Functional Selectivity, Medicine +7

RP 73870, a gastrin/cholecystokinin-B receptor antagonist with potent anti-ulcer activity in the rat.

Charles Pendley, Leo R. Fitzpatrick, Alison J. Capolino et al. · Journal of Pharmacology and Experimental Therapeutics · 1995 · 42 citations · Full text

Discovery and SAR study of novel dihydroquinoline containing glucocorticoid receptor ligands

Hidenori Takahashi, Younes Bekkali, Alison J. Capolino et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 35 citations

Medicinal Chemistry, Glucocorticoid Receptor Ligands, Biochemistry +10