Petr Jansa

Discovery of a Potent and Orally Bioavailable Cyclophilin Inhibitor Derived from the Sanglifehrin Macrocycle

Richard L. Mackman, Victoria A. Steadman, David K. Dean et al. · Journal of Medicinal Chemistry · 2018 · 75 citations · Full text

A novel and efficient one-pot synthesis of symmetrical diamide (bis-amidate) prodrugs of acyclic nucleoside phosphonates and evaluation of their biological activities

Petr Jansa, Ondřej Baszczyňski, Martin Dračínský et al. · European Journal of Medicinal Chemistry · 2011 · 59 citations

Combinatorial Chemistry, Medicinal Chemistry, Biochemistry +10

Discovery of Potent Cyclophilin Inhibitors Based on the Structural Simplification of Sanglifehrin A

Victoria A. Steadman, S. Pettit, Karine G. Poullennec et al. · Journal of Medicinal Chemistry · 2017 · 57 citations · Full text

Malonate-based inhibitors of mammalian serine racemase: Kinetic characterization and structure-based computational study

Barbora Vorlová, Dana Nachtigallová, Jana Jirásková-Vaníčková et al. · European Journal of Medicinal Chemistry · 2014 · 56 citations · Full text

Medicinal Chemistry, Drug Target, Biochemistry +11

Tautomerism and the Protonation/Deprotonation of Isocytosine in Liquid‐ and Solid‐States Studied by NMR Spectroscopy and Theoretical Calculations

Martin Dračínský, Petr Jansa, K. Ahonen et al. · European Journal of Organic Chemistry · 2011 · 46 citations

Nmr Spectroscopy, Chemistry, Spectra-structure Correlation +17