Gersande Léna

<i>In </i><i>S</i><i>ilico</i>-Guided Target Identification of a Scaffold-Focused Library:  1,3,5-Triazepan-2,6-diones as Novel Phospholipase A2 Inhibitors

Pascal Müller, Gersande Léna, Éric Boilard et al. · Journal of Medicinal Chemistry · 2006 · 67 citations · Full text

Drug Target, Pharmacotherapy, Human Spla2 Members +20

Dihydrofuro[3,4<i>-c</i>]pyridinones as Inhibitors of the Cytolytic Effects of the Pore-Forming Glycoprotein Perforin

Gersande Léna, Joseph A. Trapani, Vivien R. Sutton et al. · Journal of Medicinal Chemistry · 2008 · 36 citations · Full text

Pharmaceutical Science, Bioorganic Chemistry, Glycobiology +16

Exploration of a Series of 5-Arylidene-2-thioxoimidazolidin-4-ones as Inhibitors of the Cytolytic Protein Perforin

Julie A. Spicer, Gersande Léna, Dani M. Lyons et al. · Journal of Medicinal Chemistry · 2013 · 29 citations · Full text

Drug Target, Bioorganic Chemistry, Antiparasitic Agent +22

1,3,5‐Triazepan‐2,6‐diones as Structurally Diverse and Conformationally Constrained Dipeptide Mimetics: Identification of Malaria Liver Stage Inhibitors from a Small Pilot Library

Gersande Léna, Eliette Lallemand, Anne Charlotte Grüner et al. · Chemistry - A European Journal · 2006 · 19 citations

Combinatorial Chemistry, 1,3,5-Triazepane-2,6-dione System, Organic Chemistry +17

Synthetic Methods for the Preparation of Triazepandiones and Review of their Applications

Gersande Léna, Gilles Guichard · Current Organic Chemistry · 2008 · 12 citations

Combinatorial Chemistry, Medicinal Chemistry, Triazepine Skeletons +13