Jennifer Dao

Discovery of 1<i>H</i>-Pyrazol-3(2<i>H</i>)-ones as Potent and Selective Inhibitors of Protein Kinase R-like Endoplasmic Reticulum Kinase (PERK)

Adrian L. Smith, Kristin L. Andrews, Holger Beckmann et al. · Journal of Medicinal Chemistry · 2015 · 80 citations · Full text

Drug Target, Selective Inhibitors, Molecular Pharmacology +17

Kinetic characterization and identification of a novel inhibitor of hypoxia-inducible factor prolyl hydroxylase 2 using a time-resolved fluorescence resonance energy transfer-based assay technology

Jennifer Dao, Robert J. Kurzeja, Jose M. Morachis et al. · Analytical Biochemistry · 2008 · 70 citations

Novel Inhibitor, Aldehyde Dehydrogenase, Biochemistry +8

Discovery of novel hydroxy-thiazoles as HIF-α prolyl hydroxylase inhibitors: SAR, synthesis, and modeling evaluation

Christopher M. Tegley, Vellarkad N. Viswanadhan, Kaustav Biswas et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 44 citations · Full text

Medicinal Chemistry, Pharmaceutical Science, Biochemistry +11

Synthesis and structure–activity relationship of trisubstituted thiazoles as Cdc7 kinase inhibitors

Andreas Reichelt, Julie M. Bailis, Michael D. Bartberger et al. · European Journal of Medicinal Chemistry · 2014 · 31 citations · Full text

Structure–activity Relationship, Medicinal Chemistry, Cdc7 Kinase Inhibitors +9

Structure-guided design of substituted aza-benzimidazoles as potent hypoxia inducible factor-1α prolyl hydroxylase-2 inhibitors

Mike Frohn, Vellarkad N. Viswanadhan, Alexander J. Pickrell et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 25 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Biochemistry +13