Giulia Bianchini

Efficient synthesis of 2-acylquinolines based on an aza-vinylogous Povarov reaction

Giulia Bianchini, Pascual Ribelles, Diana Becerra et al. · Organic Chemistry Frontiers · 2016 · 46 citations

Diversity Oriented Synthesis, Natural Sciences, Diversity-oriented Synthesis +8

Design, synthesis and antiproliferative activity of decarbonyl luotonin analogues

Abdulrahman I. Almansour, Natarajan Arumugam, Raju Suresh Kumar et al. · European Journal of Medicinal Chemistry · 2017 · 42 citations

Medicine, Decarbonyl Luotonin Analogues, Pharmacology +2

Tetrahydroisoquinoline-Derived Urea and 2,5-Diketopiperazine Derivatives as Selective Antagonists of the Transient Receptor Potential Melastatin 8 (TRPM8) Channel Receptor and Antiprostate Cancer Agents

Luciano De Petrocellis, F.J. Arroyo, Pierangelo Orlando et al. · Journal of Medicinal Chemistry · 2016 · 31 citations · Full text

Trpm8 Inhibition, Pharmacotherapy, Heterocycle Chemistry +17

Crassiflorone derivatives that inhibit Trypanosoma brucei glyceraldehyde-3-phosphate dehydrogenase ( Tb GAPDH) and Trypanosoma cruzi trypanothione reductase ( Tc TR) and display trypanocidal activity

Elisa Uliassi, Giulia Fiorani, R. Luise Krauth‐Siegel et al. · European Journal of Medicinal Chemistry · 2017 · 31 citations · Full text

Tc Tr, Tb Gapdh, Biochemistry +9

B-Ring-Aryl Substituted Luotonin A Analogues with a New Binding Mode to the Topoisomerase 1-DNA Complex Show Enhanced Cytotoxic Activity

Víctor González‐Ruiz, Irene Pascua, Tamara Fernández‐Marcelo et al. · PLoS ONE · 2014 · 23 citations · Full text

Chemoprevention Strategy, Molecular Biology, Pharmacotherapy +18