Tom Willemse

The Suzuki–Miyaura Cross-Coupling as a Versatile Tool for Peptide Diversification and Cyclization

Tom Willemse, Wim Schepens, Herman van Vlijmen et al. · Catalysts · 2017 · 82 citations · Full text

Natural Sciences, Chemistry, Medicinal Chemistry +15

The First One-Pot Synthesis of <scp>l</scp>-7-Iodotryptophan from 7-Iodoindole and Serine, and an Improved Synthesis of Other <scp>l</scp>-7-Halotryptophans

Duncan R. M. Smith, Tom Willemse, Danai S. Gkotsi et al. · Organic Letters · 2014 · 62 citations

Pharmacy, Biochemistry, Medicinal Chemistry +3

A bifunctional-biased mu-opioid agonist–neuropeptide FF receptor antagonist as analgesic with improved acute and chronic side effects

Armand Drieu la Rochelle, Karel Guillemyn, Maria Dumitrascuta et al. · Pain · 2018 · 42 citations

Medicine, Medicinal Chemistry, Pharmacology +17

Suzuki–Miyaura Diversification of Amino Acids and Dipeptides in Aqueous Media

Tom Willemse, Karolien Van Imp, Rebecca J. M. Goss et al. · ChemCatChem · 2015 · 35 citations · Full text

Pharmacy, Chemical Biology, Medicinal Chemistry +15

Bromotryptophans and their incorporation in cyclic and bicyclic privileged peptides

Júlia García‐Pindado, Tom Willemse, Rebecca J. M. Goss et al. · Biopolymers · 2018 · 13 citations

Pharmacy, Chemistry, Medicinal Chemistry +17