Wim Schepens

Potent peptidic fusion inhibitors of influenza virus

Rameshwar U. Kadam, Jarek Juraszek, Boerries Brandenburg et al. · Science · 2017 · 166 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17

A small-molecule fusion inhibitor of influenza virus is orally active in mice

Maria J. P. van Dongen, Rameshwar U. Kadam, Jarek Juraszek et al. · Science · 2019 · 146 citations

Pharmacy, Infectious Diseases, Medicinal Chemistry +17

The Suzuki–Miyaura Cross-Coupling as a Versatile Tool for Peptide Diversification and Cyclization

Tom Willemse, Wim Schepens, Herman van Vlijmen et al. · Catalysts · 2017 · 82 citations · Full text

Natural Sciences, Chemistry, Medicinal Chemistry +15

The First One-Pot Synthesis of <scp>l</scp>-7-Iodotryptophan from 7-Iodoindole and Serine, and an Improved Synthesis of Other <scp>l</scp>-7-Halotryptophans

Duncan R. M. Smith, Tom Willemse, Danai S. Gkotsi et al. · Organic Letters · 2014 · 62 citations

Pharmacy, Biochemistry, Medicinal Chemistry +3

Benzoxazole and benzothiazole amides as novel pharmacokinetic enhancers of HIV protease inhibitors

Tim H. M. Jonckers, M.C. Rouan, Geerwin Haché et al. · Bioorganic & Medicinal Chemistry Letters · 2012 · 36 citations · Full text

Medicine, Pharmacokinetics, Pharmacology +15