Jozef Van Gelder

Potent and selective inhibition of HIV-1 replication in vitro by a novel series of TIBO derivatives

Rudi Pauwels, Koen Andries, Jan Desmyter et al. · Nature · 1990 · 754 citations

Selective Inhibition, Medicinal Chemistry, Medicine +11

Synthesis and anti-HIV-1 activity of 4,5,6,7-tetrahydro-5-methylimidazo[4,5,1-jk][1,4]benzodiazepin-2(1H)-one (TIBO) derivatives

Michael J. Kukla, Henry J. Breslin, Rudi Pauwels et al. · Journal of Medicinal Chemistry · 1991 · 92 citations

R 76713, a new specific non-steroidal aromatase inhibitor

Walter Wouters, R. De Coster, Marita D.W.G. Krekels et al. · Journal of Steroid Biochemistry · 1989 · 86 citations

R 76713, Biochemistry, Medicine +6

Comparative effects of the aromatase inhibitor R76713 and of its enantiomers R83839 and R83842 on steroid biosynthesis in vitro and in vivo

Walter Wouters, R. De Coster, Jacky Van Dun et al. · The Journal of Steroid Biochemistry and Molecular Biology · 1990 · 36 citations

Biosynthesis, Aromatase Inhibitor R76713, Biochemistry +9