Synthesis and evaluation of novel fluorinated pyrazolo-1,2,3-triazole hybrids as antimycobacterial agents

A Stepwise Huisgen Cycloaddition Process: Copper(I)-Catalyzed Regioselective “Ligation” of Azides and Terminal Alkynes

Vsevolod V. Rostovtsev, Luke G. Green, Valery V. Fokin et al. · Angewandte Chemie International Edition · 2002 · 11.5K citations

Natural Sciences, Chemistry, Catalysis +8

Copper(I)-Catalyzed Synthesis of Azoles. DFT Study Predicts Unprecedented Reactivity and Intermediates

Fahmi Himo, Timothy Lovell, Robert Hilgraf et al. · Journal of the American Chemical Society · 2004 · 1.7K citations

Natural Sciences, Chemistry, Medicinal Chemistry +16

1,2,3‐Triazole as a Peptide Surrogate in the Rapid Synthesis of HIV‐1 Protease Inhibitors

Ashraf Brik, Jerry Alexandratos, Ying‐Chuan Lin et al. · ChemBioChem · 2005 · 282 citations

Pharmacy, Medicinal Chemistry, Pharmacology +16

Targeting mycobacterium protein tyrosine phosphatase B for antituberculosis agents

Bo Zhou, Yantao He, Xian Zhang et al. · Proceedings of the National Academy of Sciences · 2010 · 245 citations · Full text

Life Sciences, Immunology, Pharmacology +17

Clubbed [1,2,3] triazoles by fluorine benzimidazole: A novel approach to H37Rv inhibitors as a potential treatment for tuberculosis

Charansingh H. Gill, Ganesh R. Jadhav, Mohammad Usman Shaikh et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 229 citations

Pharmacy, Medicinal Chemistry, Pharmacology +13