Journal of Thoracic Oncology · 2024 · 47 citations · 22 references
MedicineOncologyPharmacologyClinical PharmacologyMolecular OncologyOncology PharmacotherapyMonoclonal Antibody TherapyKras G12c InhibitionKras InhibitorsKras-targeted TherapyPivotal Study DesignRas Resistance MechanismsRas-targeted Therapies
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K-Ras(G12C) inhibitors allosterically control GTP affinity and effector interactions
J.M. Ostrem, Ulf Peters, Martin L. Sos et al. · Nature · 2013 · 2.5K citations · Full text
Nasser H. Hanna, Frances A. Shepherd, Frank V. Fossella et al. · Journal of Clinical Oncology · 2004 · 2.4K citations · Full text
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Sotorasib for Lung Cancers with <i>KRAS</i> p.G12C Mutation
Ferdinandos Skoulidis, Bob T. Li, Grace K. Dy et al. · New England Journal of Medicine · 2021 · 1.8K citations · Full text
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