Homogeneous multi-payload antibody–drug conjugates

Quantitative reactivity profiling predicts functional cysteines in proteomes

Eranthie Weerapana, Chu Wang, Gabriel M. Simon et al. · Nature · 2010 · 1.7K citations · Full text

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A General Method for Site-specific Incorporation of Unnatural Amino Acids into Proteins

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Conjugation site modulates the in vivo stability and therapeutic activity of antibody-drug conjugates

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