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PharmacyMedicinal ChemistryPharmacologyDrug DesignDrug DiscoveryOrganic ChemistryChemical Library DesignChemical Space ExplorationEnzyme InhibitionLead Compound DesignLigand-based DesignStructure-activity Relationship AnalysisCarbonic Anhydrase FunctionCarbonic Anhydrase InhibitorsCarbonic Anhydrase TargetsChemical Synthesis Of AnaloguesMedicinal Chemistry ApplicationsScaffold-based Library DesignTriazole Chemistry
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The Determination of Enzyme Dissociation Constants
Hans Lineweaver, Dean Burk · Journal of the American Chemical Society · 1934 · 12.1K citations