Synthesis and preclinical evaluation of a heterodimeric radioligand targeting fibroblast activation protein and integrin-αvβ3

⁶⁸Ga-FAPI PET/CT: Tracer Uptake in 28 Different Kinds of Cancer

Clemens Kratochwil, Paul Flechsig, Thomas Lindner et al. · Journal of Nuclear Medicine · 2019 · 1.4K citations · Full text

Medicine, Nuclear Medicine, Oncology +17

A Tumor-Imaging Method Targeting Cancer-Associated Fibroblasts

Anastasia Loktev, Thomas Lindner, Walter Mier et al. · Journal of Nuclear Medicine · 2018 · 770 citations · Full text

Medicine, Nuclear Medicine, Oncology +17

Comparison of [68Ga]Ga-DOTA-FAPI-04 and [18F] FDG PET/CT for the diagnosis of primary and metastatic lesions in patients with various types of cancer

Haojun Chen, Yizhen Pang, Jingxun Wu et al. · European Journal of Nuclear Medicine and Molecular Imaging · 2020 · 540 citations

Medicine, Oncology, Radiology +12

FAPI-74 PET/CT Using Either¹⁸F-AlF or Cold-Kit⁶⁸Ga Labeling: Biodistribution, Radiation Dosimetry, and Tumor Delineation in Lung Cancer Patients

Frederik L. Giesel, Sebastian Adeberg, Mustafa Syed et al. · Journal of Nuclear Medicine · 2020 · 303 citations · Full text

Medicine, Nuclear Medicine, Oncology +17

Selective Inhibitors of Fibroblast Activation Protein (FAP) with a (4-Quinolinoyl)-glycyl-2-cyanopyrrolidine Scaffold

Koen Jansen, Leen Heirbaut, Jonathan D. Cheng et al. · ACS Medicinal Chemistry Letters · 2013 · 260 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +11