Concepedia

Development and structure-activity relationship of tacrine derivatives as highly potent CDK2/9 inhibitors for the treatment of cancer

Limeng Wu, Wenjie Liu, Wenjie Liu, Yaoguang Huang, Chengze Zhu, Qun Ma, Qiong Wu, Liting Tian, Xiangling Feng, Mingyue Liu,

European Journal of Medicinal Chemistry · 2022 · 13 citations · 35 references

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35

A new and rapid colorimetric determination of acetylcholinesterase activity

George L. Ellman, K. Diane Courtney, Valentino Andres et al. · Biochemical Pharmacology · 1961 · 26.9K citations

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Circ3823 contributes to growth, metastasis and angiogenesis of colorectal cancer: involvement of miR-30c-5p/TCF7 axis

Yaxin Guo, Yuying Guo, Chen Chen et al. · Molecular Cancer · 2021 · 223 citations · Full text

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Cyclin Dependent Kinase 9 Inhibitors for Cancer Therapy

Yogesh A. Sonawane, Margaret Taylor, John V. Napoleon et al. · Journal of Medicinal Chemistry · 2016 · 153 citations · Full text

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Discovery of PF-06873600, a CDK2/4/6 Inhibitor for the Treatment of Cancer

Kevin D. Freeman‐Cook, Robert L. Hoffman, Douglas C. Behenna et al. · Journal of Medicinal Chemistry · 2021 · 117 citations · Full text

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Development of selective mono or dual PROTAC degrader probe of CDK isoforms

Fei Zhou, Luyu Chen, Chao-Guo Cao et al. · European Journal of Medicinal Chemistry · 2019 · 107 citations · Full text

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