Concepedia

Novel structural hybrids of quinoline and thiazole moieties: Synthesis and evaluation of antibacterial and antifungal activities with molecular modeling studies

Sally I. Eissa, Amel M. Farrag, Samir Y. Abbas, Mohamed F. El Shehry, Ahmed Ragab, Eman A. Fayed, Yousry A. Ammar

Bioorganic Chemistry · 2021 · 110 citations · 35 references

DOI

Concepts

References

35

SwissADME: a free web tool to evaluate pharmacokinetics, drug-likeness and medicinal chemistry friendliness of small molecules

Antoine Daina, Olivier Michielin, Vincent Zoete · Scientific Reports · 2017 · 17.1K citations · Full text

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Phenethylthiazolethiourea (PETT) Compounds, a New Class of HIV-1 Reverse Transcriptase Inhibitors. 1. Synthesis and Basic Structure-Activity Relationship Studies of PETT Analogs

Frank W. Bell, Amanda Cantrell, Marita Hoegberg et al. · Journal of Medicinal Chemistry · 1995 · 455 citations · Full text

, , +15

Quinoline: A versatile heterocyclic

Akranth Marella, Omprakash Tanwar, Rikta Saha et al. · Saudi Pharmaceutical Journal · 2012 · 447 citations · Full text

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Structure-activity relationships of a series of 2-amino-4-thiazole-containing renin inhibitors

William C. Patt, Harriet W. Hamilton, Michael D. Taylor et al. · Journal of Medicinal Chemistry · 1992 · 373 citations · Full text

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N-(4-Substituted-thiazolyl)oxamic acid derivatives, new series of potent, orally active antiallergy agents

Karl D. Hargrave, Friedrich K. Hess, James T. Oliver · Journal of Medicinal Chemistry · 1983 · 321 citations

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