Discovery of novel steroidal-chalcone hybrids with potent and selective activity against triple-negative breast cancer

Anti-HIV-1 protease activity of compounds from Boesenbergia pandurata

Sarot Cheenpracha, Chatchanok Karalai, Chanita Ponglimanont et al. · Bioorganic & Medicinal Chemistry · 2005 · 233 citations

Medicinal Chemistry, Biochemistry, Natural Sciences +5

The Discovery of Polo-Like Kinase 4 Inhibitors: Identification of (1<i>R</i>,2<i>S</i>)-2-(3-((<i>E</i>)-4-(((<i>cis</i>)-2,6-Dimethylmorpholino)methyl)styryl)-1<i>H</i>-indazol-6-yl)-5′-methoxyspiro[cyclopropane-1,3′-indolin]-2′-one (CFI-400945) as a Potent, Orally Active Antitumor Agent

Peter B. Sampson, Yong Liu, Bryan Forrest et al. · Journal of Medicinal Chemistry · 2014 · 166 citations · Full text

Studies on novel D-ring substituted steroidal pyrazolines as potential anticancer agents

Abid H. Banday, Bilal P. Mir, Imtiyaz H. Lone et al. · Steroids · 2010 · 140 citations

Medicinal Chemistry, Novel D-ring, Steroidal Pyrazolines +9

Isatin Derived Spirocyclic Analogues with α-Methylene-γ-butyrolactone as Anticancer Agents: A Structure–Activity Relationship Study

Sandeep Rana, Elizabeth C. Blowers, Calvin Tebbe et al. · Journal of Medicinal Chemistry · 2016 · 111 citations · Full text

Chemoprevention Strategy, Pharmacotherapy, Anticancer Agents +20

Efficient synthesis of new antiproliferative steroidal hybrids using the molecular hybridization approach

Bin Yu, Ping‐Ping Qi, Xiaojing Shi et al. · European Journal of Medicinal Chemistry · 2016 · 82 citations · Full text

Combinatorial Chemistry, Engineering, Medicine +11