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PharmacyMedicinal ChemistryPharmacologyDrug DesignDrug DiscoveryStructure-activity RelationshipsAntibacterial AgentsAntibacterial PharmacologyAntimicrobial PeptidesPeptidomimetic DesignAbsolute Configuration AssignmentAbsolute Configuration DeterminationAntibiotic DiscoveryNovel Antibacterial Drug DiscoveryPeptide Structure-activity RelationshipsSelectivitySelectivity Index Optimization
, paired with favorable selectivity (selectivity index >60), which collectively underscores the promise of the rufomycins as potential anti-TB drug leads.
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