Concepedia

Identification of novel GPR81 agonist lead series for target biology evaluation

Öjvind Davidsson, Kristina Nilsson, Jonas Brånalt, Terese Andersson, Kristina Berggren, Yantao Chen, Ola Fjellström, Henrik Gradén, Linda Gustafsson, Nils-Olov Hermansson,

Bioorganic & Medicinal Chemistry Letters · 2020 · 11 citations · 26 references

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26

The Cambridge Structural Database: a quarter of a million crystal structures and rising

Frank H. Allen · Acta Crystallographica Section B Structural Science · 2002 · 10.3K citations

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PUMA-G and HM74 are receptors for nicotinic acid and mediate its anti-lipolytic effect

Sorin Tunaru, Jukka Kero, Annette Schaub et al. · Nature Medicine · 2003 · 795 citations

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Lactate Inhibits Lipolysis in Fat Cells through Activation of an Orphan G-protein-coupled Receptor, GPR81

Changlu Liu, Jiejun Wu, Jessica Zhu et al. · Journal of Biological Chemistry · 2008 · 589 citations · Full text

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Molecular Identification of High and Low Affinity Receptors for Nicotinic Acid

Alan Wise, Steven M. Foord, Neil J. Fraser et al. · Journal of Biological Chemistry · 2003 · 541 citations · Full text

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An Autocrine Lactate Loop Mediates Insulin-Dependent Inhibition of Lipolysis through GPR81

Kashan Ahmed, Sorin Tunaru, Cong Tang et al. · Cell Metabolism · 2010 · 443 citations · Full text

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