Design, synthesis, and structure-activity relationship studies of novel triazole agents with strong antifungal activity against Aspergillus fumigatus

Structural analyses of Candida albicans sterol 14α-demethylase complexed with azole drugs address the molecular basis of azole-mediated inhibition of fungal sterol biosynthesis

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Life Sciences, Biochemistry, Pharmacology +17

New Azole Antifungals. 3. Synthesis and Antifungal Activity of 3-Substituted-4(3<i>H</i>)-quinazolinones

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Yeast cytochrome P-450 catalyzing lanosterol 14 alpha-demethylation. II. Lanosterol metabolism by purified P-450(14)DM and by intact microsomes.

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Life Sciences, Biochemistry, Molecular Biology +16

Structure-Functional Characterization of Cytochrome P450 Sterol 14α-Demethylase (CYP51B) from Aspergillus fumigatus and Molecular Basis for the Development of Antifungal Drugs

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Medicine, Molecular Biology, Pharmacology +17

Design, Synthesis, and Structure–Activity Relationship Studies of Novel Fused Heterocycles-Linked Triazoles with Good Activity and Water Solubility

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Pharmacy, Medicinal Chemistry, Pharmacology +17