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Catalytic C(sp3)–H bond activation in tertiary alkylamines

Jesus Rodrigalvarez, Manuel Nappi, Hiroki Azuma, Nils J. Flodén, Matthew Burns, Matthew J. Gaunt

Nature Chemistry · 2019 · 111 citations · 37 references

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37

The Medicinal Chemist’s Toolbox: An Analysis of Reactions Used in the Pursuit of Drug Candidates

Stephen D. Roughley, Allan M. Jordan · Journal of Medicinal Chemistry · 2011 · 2.7K citations

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Catalytic Functionalization of C(sp<sup>2</sup>)H and C(sp<sup>3</sup>)H Bonds by Using Bidentate Directing Groups

Guy Rouquet, Naoto Chatani · Angewandte Chemie International Edition · 2013 · 2K citations

, , +13

Highly Regioselective Arylation of sp<sup>3</sup> C−H Bonds Catalyzed by Palladium Acetate

V. G. Zaitsev, Dmitry Shabashov, Olafs Daugulis · Journal of the American Chemical Society · 2005 · 1.5K citations

, , +13

Palladium-Catalyzed Methylation and Arylation of sp<sup>2</sup> and sp<sup>3</sup> C−H Bonds in Simple Carboxylic Acids

Ramesh Giri, Nathan Maugel, Jiao-Jie Li et al. · Journal of the American Chemical Society · 2007 · 773 citations

, , +16

Knowledge-Based, Central Nervous System (CNS) Lead Selection and Lead Optimization for CNS Drug Discovery

Arup K. Ghose, Torsten Herbertz, Robert L. Hudkins et al. · ACS Chemical Neuroscience · 2011 · 437 citations · Full text

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