Organic Chemistry Frontiers · 2019 · 14 citations · 28 references
PharmacyMolecular PharmaceuticsPharmaceuticsAntibody EngineeringDrug DeliveryStructural BiologyAntibody ConjugatesAntibody ConjugationAntibody StabilityAntibody StructureAntibody-antigen RecognitionAntibody-drug ConjugatesAntibody Glycosylation ControlAntibody Glycosylation EffectsAntibody-drug Conjugate LinkersAntibody-drug LinkersConjugate CharacterizationConjugationConjugation Chemistry For AntibodiesGlycoengineering Of Monoclonal Antibodies
Two new linkers employed in glycosite-specific antibody–drug conjugates demonstrate efficient conjugation, enhanced stability, and fluorescence properties.
28
Development of potent monoclonal antibody auristatin conjugates for cancer therapy
Svetlana O. Doronina, Brian E. Toki, Michael Torgov et al. · Nature Biotechnology · 2003 · 1.2K citations