Concepedia

Synthesis and sar of 4-(1H-benzimidazole-2-carbonyl)piperidines with dual histamine H1/tachykinin NK1 receptor antagonist activity

George D. Maynard, Larry Bratton, John M. Kane, Timothy P. Burkholder, Braulio Santiago, Kenneth T. Stewart, Elizabeth M. Kudlacz, Scott A. Shatzer, Robert W. Knippenberg, Amy M. Farrell,

Bioorganic & Medicinal Chemistry Letters · 1997 · 16 citations · 3 references

DOI

Concepts

References

3

The Use of Diethyl Azodicarboxylate and Triphenylphosphine in Synthesis and Transformation of Natural Products

Oyo Mitsunobu · Synthesis · 1981 · 4.1K citations

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Identification and chemical synthesis of MDL 105,212, a non-peptide tachykinin antagonist with high affinity for NK1 and NK2 receptors

Timothy P. Burkholder, Elizabeth M. Kudlacz, Tieu-Binh Le et al. · Bioorganic & Medicinal Chemistry Letters · 1996 · 29 citations

, , +6

A highly convergent synthesis of benzimidazolylpiperidines

Albert A. Carr, David Hay, John M. Kane et al. · The Journal of Organic Chemistry · 1990 · 10 citations

, , +7