Efficient synthesis of imidazopyridodiazepines from peri annulation in imidazo[1,2-a]pyridine

Synthesis and anti-HIV-1 activity of 4,5,6,7-tetrahydro-5-methylimidazo[4,5,1-jk][1,4]benzodiazepin-2(1H)-one (TIBO) derivatives. 2

Michael J. Kukla, Henry J. Breslin, Craig J. Diamond et al. · Journal of Medicinal Chemistry · 1991 · 166 citations

Pharmacy, Chemistry, Medicinal Chemistry +12

Study of the Pictet-Spengler reaction in aprotic media: synthesis of the .beta.-galactosidase inhibitor, pyridindolol

Dave Soerens, J. SANDRIN, F. UNGEMACH et al. · The Journal of Organic Chemistry · 1979 · 134 citations

Life Sciences, Biochemistry, Chemistry +5

General method for the assignment of stereochemistry of 1,3-disubstituted 1,2,3,4-tetrahydro-.beta.-carbolines by carbon-13 spectroscopy

F. UNGEMACH, Dave Soerens, Richard W. Weber et al. · Journal of the American Chemical Society · 1980 · 104 citations

Natural Sciences, Chemistry, Medicinal Chemistry +7

Electrophilic substitution in indoles—IV

A. H. JACKSON, Balakrishna Naidoo, Paul E. Smith · Tetrahedron · 1968 · 98 citations

Natural Sciences, Chemistry, Medicinal Chemistry +6

Synthesis and Anti-HIV-1 Activity of 4,5,6,7-Tetrahydro-5-methylimidazo[4,5,1-jk][1,4]benzodiazepin-2(1H)-one (TIBO) Derivatives. 3

Henry J. Breslin, Michael J. Kukla, Donald Ludovici et al. · Journal of Medicinal Chemistry · 1995 · 97 citations

Pharmacy, Medicinal Chemistry, Pharmacology +6