Concepedia

A novel trifluoromethanesulfonamidophenyl-substituted quinoline derivative, GA 0113: synthesis and pharmacological profiles

Yoshitomi Morizawa, Takashi Okazoe, Shu‐zhong Wang, Junichi Sasaki, Hajime Ebisu, Masakuni Nishikawa, Hiroshi Shinyama

Journal of Fluorine Chemistry · 2001 · 34 citations · 6 references

DOI

Concepts

References

6

The discovery of potent nonpeptide angiotensin II receptor antagonists: a new class of potent antihypertensives

John V. Duncia, Andrew T. Chiu, David J. Carini et al. · Journal of Medicinal Chemistry · 1990 · 241 citations · Full text

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Nonpeptide angiotensin II receptor antagonists. Synthesis and biological activity of potential prodrugs of benzimidazole-7-carboxylic acids

Yasuhisa Kohara, Y. Yoshimura, Yumiko Shibouta et al. · Journal of Medicinal Chemistry · 1993 · 129 citations

, , +13

Sulfonylureas and Sulfonylcarbamates as New Non-Tetrazole Angiotensin II Receptor Antagonists. Discovery of a Highly Potent Orally Active (Imidazolylbiphenylyl)sulfonylurea (HR 720)

Pierre Deprez, Jacques Guillaume, R. H. A. Becker et al. · Journal of Medicinal Chemistry · 1995 · 64 citations · Full text

, , +9

Triazolinone Biphenylsulfonamide Derivatives as Orally Active Angiotensin II Antagonists with Potent AT1 Receptor Affinity and Enhanced AT2 Affinity

Wallace T. Ashton, Linda Chang, Kelly L. Flanagan et al. · Journal of Medicinal Chemistry · 1994 · 37 citations · Full text

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Pharmacologic Profiles of GA0113, a Novel Quinoline Derivative Angiotensin II AT1-Receptor Antagonist

Hajime Ebisu, Masakuni Nishikawa, Mikio Tanaka et al. · Journal of Cardiovascular Pharmacology · 1999 · 25 citations

, , +17