Stereochemically controlled syntheses of indole-substituted dihydrofuran-2-ones and a pyrrolidin-2-one

Pharmacophore/Receptor Models for GABA_A/BzR Subtypes (α1β3γ2, α5β3γ2, and α6β3γ2) via a Comprehensive Ligand-Mapping Approach

Qi Huang, Xiaohui He, Chunrong Ma et al. · Journal of Medicinal Chemistry · 1999 · 135 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

A Convenient Synthesis of Conformationally Constrained β-Substituted Tryptophans

Csaba Nemes, Laurent Jeannin, János Sápi et al. · Tetrahedron · 2000 · 67 citations

Natural Sciences, Biochemistry, Chemistry +6

Improved Synthesis of Isogranulatimide, a G2 Checkpoint Inhibitor. Syntheses of Didemnimide C, Isodidemnimide A, Neodidemnimide A, 17-Methylgranulatimide, and Isogranulatimides A−C

Edward Piers, Robert Britton, Raymond J. Andersen · The Journal of Organic Chemistry · 1999 · 60 citations

Pharmacy, Medicinal Chemistry, Pharmacology +11

Synthesis and cyclisation of didemnimide C and its imidazol-1-yl isomer

Andreas Terpin, Christian Winklhofer, Susanne Schumann et al. · Tetrahedron · 1998 · 46 citations

Natural Sciences, Chemistry, Medicinal Chemistry +8

1,3-Dipolar Cycloadditions of Diazomethane to Chiral Electron-Deficient Olefins:  The Origin of the π-Facial Diastereoselection

Elena Muray, Ángel Álvarez‐Larena, J.F. Piniella et al. · The Journal of Organic Chemistry · 1999 · 37 citations

Natural Sciences, Chemistry, Organic Chemistry +8