Concepedia

Defined concatenated α6α1β3γ2 GABAA receptor constructs reveal dual action of pyrazoloquinolinone allosteric modulators

Xenia Simeone, M.T. Iorio, David Chan Bodin Siebert, Sabah Rehman, Michael Schnürch, Marko D. Mihovilovič, Margot Ernst

Bioorganic & Medicinal Chemistry · 2019 · 14 citations · 34 references

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GABAA receptors: immunocytochemical distribution of 13 subunits in the adult rat brain

Susanne Pirker, Christoph Schwarzer, Anna Wieselthaler et al. · Neuroscience · 2000 · 1.3K citations

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Segregation of Different GABA<sub>A</sub>Receptors to Synaptic and Extrasynaptic Membranes of Cerebellar Granule Cells

Zoltán Nusser, Werner Sieghart, Péter Somogyi · Journal of Neuroscience · 1998 · 835 citations · Full text

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Structure of a human synaptic GABAA receptor

Shaotong Zhu, Colleen Noviello, Jinfeng Teng et al. · Nature · 2018 · 569 citations · Full text

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GABAA receptor signalling mechanisms revealed by structural pharmacology

Simonas Masiulis, Rooma Desai, Tomasz Uchański et al. · Nature · 2018 · 557 citations

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Forced Subunit Assembly in α1β2γ2 GABAAReceptors

Sabine W. Baumann, Roland Baur, Erwin Sigel · Journal of Biological Chemistry · 2002 · 260 citations · Full text

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