Concepedia

Identification of a new tamoxifen-xanthene hybrid as pro-apoptotic anticancer agent

Elena Catanzaro, Francesca Seghetti, Cinzia Calcabrini, Angela Rampa, Silvia Gobbi, Piero Sestili, Eleonora Turrini, Francesca Maffei, Patrizia Hrelia, Alessandra Bisi,

Bioorganic Chemistry · 2019 · 28 citations · 25 references

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25

Down-regulation of bcl-2 by p53 in breast cancer cells.

Subrata Haldar, Massimo Negrini, Maria Monne et al. · PubMed · 1994 · 479 citations

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Genotoxic potential of tamoxifen and analogues in female Fischer F344/n rats, DBA/2 and C57BL/6 mice and in human MCL-5 cells

Ian N.H. White, Adrian Davies, Lewis L. Smith et al. · Carcinogenesis · 1992 · 239 citations

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Activation of caspase-3 and c-Jun NH2-terminal kinase-1 signaling pathways in tamoxifen-induced apoptosis of human breast cancer cells.

Sandhya Mandlekar, Rong Yu, Tse‐Hua Tan et al. · PubMed · 2000 · 199 citations

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Tamoxifen antiestrogens. A comparison of the activity, pharmacokinetics, and metabolic activation of the cis and trans isomers of tamoxifen

David W. Robertson, John A. Katzenellenbogen, Deborah J. Long et al. · Journal of Steroid Biochemistry · 1982 · 171 citations

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Differential sensitivity of human breast cancer cell lines to the growth-inhibitory effects of tamoxifen.

Roger R. Reddel, Leigh C. Murphy, Rosemary E. Hall et al. · PubMed · 1985 · 170 citations

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