Concepedia

Belinostat, at Its Clinically Relevant Concentrations, Inhibits Rifampicin-Induced CYP3A4 and MDR1 Gene Expression

Kodye L. Abbott, Chloe S. Chaudhury, Aneesh Chandran, Saraswathi Vishveshwara, Zdeněk Dvořák, Eva Jiskrová, Karolína Poulíková, Barbora Vyhlídalová, Sridhar Mani, Satyanarayana R. Pondugula

Molecular Pharmacology · 2019 · 16 citations · 40 references

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40

Development and validation of a genetic algorithm for flexible docking 1 1Edited by F. E. Cohen

Gareth Jones, Peter Willett, Robert C. Glen et al. · Journal of Molecular Biology · 1997 · 6.7K citations

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The orphan nuclear receptor SXR coordinately regulates drug metabolism and efflux

Timothy W. Synold, Isabelle Dussault, Barry M. Forman · Nature Medicine · 2001 · 834 citations

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CYP3A4 Induction by Drugs: Correlation between a Pregnane X Receptor Reporter Gene Assay and CYP3A4 Expression in Human Hepatocytes

Gang Luo, Mark R. Cunningham, Sean Kim et al. · Drug Metabolism and Disposition · 2002 · 447 citations

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Dexamethasone Induces Pregnane X Receptor and Retinoid X Receptor-α Expression in Human Hepatocytes: Synergistic Increase of CYP3A4 Induction by Pregnane X Receptor Activators

Jean‐Marc Pascussi, Lionel Drocourt, Jean‐Michel Fabre et al. · Molecular Pharmacology · 2000 · 367 citations

, , +11

Dual effect of dexamethasone on <i>CYP3A4</i> gene expression in human hepatocytes

Jean‐Marc Pascussi, Lionel Drocourt, Sabine Gerbal‐Chaloin et al. · European Journal of Biochemistry · 2001 · 299 citations · Full text

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