Concepedia

Synthesis, biological evaluation, and molecular modeling of 11H-indeno[1,2-b]quinoxalin-11-one derivatives and tryptanthrin-6-oxime as c-Jun N-terminal kinase inhibitors

Igor A. Schepetkin, Аndrei I. Khlebnikov, Аndrei S. Potapov, Anastasia R. Kovrizhina, Vladislava V. Matveevskaya, M. L. Belyanin, Dmitriy N. Atochin, Svitlana O. Zanoza, Nadiya M. Gaidarzhy, S. А. Lyakhov,

European Journal of Medicinal Chemistry · 2018 · 80 citations · 45 references

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References

45

A quantitative analysis of kinase inhibitor selectivity

Mazen W. Karaman, Sanna Herrgård, Daniel K. Treiber et al. · Nature Biotechnology · 2008 · 2.4K citations

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A small molecule–kinase interaction map for clinical kinase inhibitors

Miles A. Fabian, William Biggs, Daniel K. Treiber et al. · Nature Biotechnology · 2005 · 1.9K citations · Full text

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The specificities of protein kinase inhibitors: an update

Jenny Bain, Hilary McLauchlan, Matthew Elliott et al. · Biochemical Journal · 2003 · 1.4K citations · Full text

, , +11

Selective interaction of JNK protein kinase isoforms with transcription factors.

Shreyasi Gupta, Tyler W. Barrett, Alan J. Whitmarsh et al. · The EMBO Journal · 1996 · 1.3K citations · Full text

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Discovery of Tryptanthrin Derivatives as Potent Inhibitors of Indoleamine 2,3-Dioxygenase with Therapeutic Activity in Lewis Lung Cancer (LLC) Tumor-Bearing Mice

Shuangshuang Yang, Xishuai Li, Fangfang Hu et al. · Journal of Medicinal Chemistry · 2013 · 181 citations · Full text

, , +15