Concepedia

Design and synthesis of functionalized piperazin-1yl-(E)-stilbenes as inhibitors of 17α-hydroxylase-C17,20-lyase (Cyp17)

Benjamin E. Blass, Pravin S. Iyer, Magid Abou‐Gharbia, Wayne E. Childers, John Gordon, Mercy Ramanjulu, George Morton, Premkumar Arumugam, Joshodeep Boruwa, John W. Ellingboe,

Bioorganic & Medicinal Chemistry Letters · 2018 · 12 citations · 3 references

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Novel Steroidal Inhibitors of Human Cytochrome P45017.alpha.-Hydroxylase-C17,20-lyase): Potential Agents for the Treatment of Prostatic Cancer

Gerard A. Potter, S. Elaine Barrie, Michael Jarman et al. · Journal of Medicinal Chemistry · 1995 · 380 citations · Full text

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Highly-selective 4-(1,2,3-triazole)-based P450c17a 17,20-lyase inhibitors

Stephen W Rafferty, Joel R. Eisner, William R. Moore et al. · Bioorganic & Medicinal Chemistry Letters · 2014 · 57 citations · Full text

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Design, synthesis, and evaluation of (2S,4R)-Ketoconazole sulfonamide analogs as potential treatments for Metabolic Syndrome

Benjamin E. Blass, Pravin S. Iyer, Magid Abou‐Gharbia et al. · Bioorganic & Medicinal Chemistry Letters · 2016 · 13 citations · Full text

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