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Evaluation of sulphonamide derivatives acting as inhibitors of human carbonic anhydrase isoforms I, II and<i>Mycobacterium tuberculosis</i><b>β</b>-class enzyme Rv3273

Tanvi V. Wani, Silvia Bua, Pravin S. Khude, Abdul H. Chowdhary, Claudiu T. Supuran, Mrunmayee P. Toraskar

Journal of Enzyme Inhibition and Medicinal Chemistry · 2018 · 33 citations · 15 references

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Abstract

s were in the range of 54.6 nM-1.8 µM against hCA I, in the range of 32.1 nM-5.5 µM against hCA II and of 127 nM-2.12 µM against mtCA 3.

References

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