Concepedia

Design, synthesis, and biological evaluation of novel combretastatin A-4 thio derivatives as microtubule targeting agents

Tomasz Stefański, Renata Mikstacka, Rafał Kurczab, Zbigniew Dutkiewicz, Małgorzata Kucińska, Marek Murias, Małgorzata Zielińska‐Przyjemska, Michał Cichocki, Anna Teubert, Mariusz Kaczmarek,

European Journal of Medicinal Chemistry · 2017 · 31 citations · 41 references

DOI

Concepts

References

41

Directory of Useful Decoys, Enhanced (DUD-E): Better Ligands and Decoys for Better Benchmarking

Michael M. Mysinger, Michael Carchia, John J. Irwin et al. · Journal of Medicinal Chemistry · 2012 · 2.4K citations · Full text

, , +17

Structure of the αβ tubulin dimer by electron crystallography

Eva Nogales, Sharon G. Wolf, Kenneth H. Downing · Nature · 1998 · 2.1K citations

, , +13

Insight into tubulin regulation from a complex with colchicine and a stathmin-like domain

Raimond B. G. Ravelli, Benoı̂t Gigant, Patrick A. Curmi et al. · Nature · 2004 · 1.6K citations

, , +14

Isolation and structure of the strong cell growth and tubulin inhibitor combretastatin A-4

George R. Pettit, Sheo B. Singh, Ernest Hamel et al. · Cellular and Molecular Life Sciences · 1989 · 789 citations

, , +11

Structural basis for the regulation of tubulin by vinblastine

Benoı̂t Gigant, Chunguang Wang, Raimond B. G. Ravelli et al. · Nature · 2005 · 730 citations

, , +11