Concepedia

A comparative study of amide-bond forming reagents in aqueous media – Substrate scope and reagent compatibility

Matthew Badland, Robert Crook, Bastien Delayre, Steven J. Fussell, Iain R. Gladwell, Michael Hawksworth, Roger M. Howard, Robert Walton, Gerald A. Weisenburger

Tetrahedron Letters · 2017 · 40 citations · 23 references

DOI

Concepts

References

23

Analysis of Past and Present Synthetic Methodologies on Medicinal Chemistry: Where Have All the New Reactions Gone?

Dean G. Brown, Jonas Boström · Journal of Medicinal Chemistry · 2015 · 2K citations · Full text

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Amide bond formation and peptide coupling

Christian Montalbetti, Virginie M. Falque · Tetrahedron · 2005 · 1.7K citations

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Large-Scale Applications of Amide Coupling Reagents for the Synthesis of Pharmaceuticals

Joshua R. Dunetz, Javier Magano, Gerald A. Weisenburger · Organic Process Research & Development · 2015 · 799 citations

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Mechanism of Amide Formation by Carbodiimide for Bioconjugation in Aqueous Media

Naoki Nakajima, Yoshito Ikada · Bioconjugate Chemistry · 1995 · 761 citations

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Formation of carboxamides by direct condensation of carboxylic acids and amines in alcohols using a new alcohol- and water-soluble condensing agent: DMT-MM

Munetaka Kunishima, Chiho Kawachi, Kazuhito Hioki et al. · Tetrahedron · 2001 · 344 citations

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