Concepedia

Imidazo[1,2-a]pyrazine, Imidazo[1,5-a]quinoxaline and Pyrazolo[1,5-a]quinoxaline derivatives as IKK1 and IKK2 inhibitors

Cindy Patinote, Nour Bou Karroum, Georges Moarbess, Carine Deleuze‐Masquéfa, Kamel Hadj‐Kaddour, Pierre Cuq, Mona Diab‐Assaf, Issam Kassab, Pierre‐Antoine Bonnet

European Journal of Medicinal Chemistry · 2017 · 30 citations · 16 references

DOI

Concepts

References

16

Inhibition of NF-κB by Sodium Salicylate and Aspirin

Elizabeth B. Kopp, Sankar Ghosh · Science · 1994 · 1.8K citations

, , +17

The anti-inflammatory agents aspirin and salicylate inhibit the activity of IκB kinase-β

Min-Jean Yin, Yumi Yamamoto, Richard B. Gaynor · Nature · 1998 · 1.6K citations

, , +14

Sulfasalazine: a potent and specific inhibitor of nuclear factor kappa B.

Claudia Wahl, Susanne Liptay, G. Adler et al. · Journal of Clinical Investigation · 1998 · 740 citations · Full text

, , +17

BMS-345541 Is a Highly Selective Inhibitor of IκB Kinase That Binds at an Allosteric Site of the Enzyme and Blocks NF-κB-dependent Transcription in Mice

James R. Burke, Mark A. Pattoli, Kurt R. Gregor et al. · Journal of Biological Chemistry · 2003 · 547 citations · Full text

, , +13

Mesalamine blocks tumor necrosis factor growth inhibition and nuclear factor κB activation in mouse colonocytes

G. C. Kaiser, Fang Yan, D. Brent Polk · Gastroenterology · 1999 · 232 citations · Full text

, , +16