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Synthesis and biological evaluation of fluorinated N -benzoyl and N -phenylacetoyl derivatives of 3-(4-aminophenyl)-coumarin-7- O -sulfamate as steroid sulfatase inhibitors

Mateusz Daśko, Maja Przybyłowska, Janusz Rachoń, Maciej Masłyk, Konrad Kubiński, Majus Misiak, Andrzej Składanowski, Sebastian Demkowicz

European Journal of Medicinal Chemistry · 2017 · 24 citations · 20 references

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20

AutoDock Vina: Improving the speed and accuracy of docking with a new scoring function, efficient optimization, and multithreading

Oleg Trott, Arthur J. Olson · Journal of Computational Chemistry · 2009 · 37.1K citations · Full text

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Fluorine in medicinal chemistry: Recent therapeutic applications of fluorinated small molecules

Kenneth L. Kirk · Journal of Fluorine Chemistry · 2006 · 892 citations

, , +13

Recent advances (1995–2005) in fluorinated pharmaceuticals based on natural products

Journal of Fluorine Chemistry · 2006 · 587 citations

, , +7

RECENT ADVANCES IN FLUORINATED PHARMACEUTICALS BASED ON NATURAL PRODUCTS

YU Hai-tao · Acta Academiae Medicinae Neimongol · 2006 · 483 citations

, , +13

Inactivation of Steroid Sulfatase by an Active Site-Directed Inhibitor, Estrone-3-O-Sulfamate

Atul Purohit, Gary J. Williams, Nicola M. Howarth et al. · Biochemistry · 1995 · 170 citations

, , +13