Advanced Synthesis & Catalysis · 2016 · 30 citations · 54 references
Natural SciencesChemistryCatalysisCoordination ChemistryCopper CatalysisFunctional Group ToleranceMaleimide ChemistryMaleimide FunctionalizationThiol ChemistryThiol FunctionalizationThiol-maleimide Coupling
Abstract An efficient copper(I) iodide‐catalyzed sulfenylation of maleimides and related 3‐indolylmaleimides with thiols has been developed in the presence of fluoroboric acid. Several 3‐thiomaleimides and 3‐indolyl‐4‐thiomaleimides were obtained with good yields under ligand‐free conditions. The methods are simple, practical and show good functional group tolerance. magnified image
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Scott D. McCann, Shannon S. Stahl · Accounts of Chemical Research · 2015 · 542 citations · Full text
Serena Pasquini, Claudia Mugnaini, Cristina Tintori et al. · Journal of Medicinal Chemistry · 2008 · 164 citations · Full text