Concepedia

Design and synthesis of cis-restricted benzimidazole and benzothiazole mimics of combretastatin A-4 as antimitotic agents with apoptosis inducing ability

Md. Ashraf, Thokhir Basha Shaik, M. Shaheer Malik, Riyaz Syed, Prema L. Mallipeddi, M.V.P.S. Vishnu Vardhan, Ähmed Kamal

Bioorganic & Medicinal Chemistry Letters · 2016 · 46 citations · 29 references

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29

Sulforhodamine B colorimetric assay for cytotoxicity screening

Vanicha Vichai, Kanyawim Kirtikara · Nature Protocols · 2006 · 3.7K citations

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Insight into tubulin regulation from a complex with colchicine and a stathmin-like domain

Raimond B. G. Ravelli, Benoı̂t Gigant, Patrick A. Curmi et al. · Nature · 2004 · 1.6K citations

, , +14

Isolation and structure of the strong cell growth and tubulin inhibitor combretastatin A-4

George R. Pettit, Sheo B. Singh, Ernest Hamel et al. · Cellular and Molecular Life Sciences · 1989 · 789 citations

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The microtubule-affecting drug paclitaxel has antiangiogenic activity.

Dorina Belotti, Veronica Vergani, Teresa Drudis et al. · PubMed · 1996 · 646 citations

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Antimitotic natural products combretastatin A-4 and combretastatin A-2: studies on the mechanism of their inhibition of the binding of colchicine to tubulin

Chii M. Lin, Holly H. Ho, George R. Pettit et al. · Biochemistry · 1989 · 414 citations

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