Concepedia

1,1′-Carbonyldiimidazole (CDI) Mediated Coupling and Cyclization To Generate [1,2,4]Triazolo[4,3-<i>a</i>]pyridines

Kyle D. Baucom, Siân C. Jones, Scott W. Roberts

Organic Letters · 2016 · 26 citations · 29 references

DOI

Concepts

Abstract

An operationally efficient CDI mediated tandem coupling and cyclization reaction to generate [1,2,4]triazolo[4,3-a]pyridines has been reported. The reaction conditions and scope were investigated, and the methodology was demonstrated in batch mode as well as in a continuous process.

References

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