The Journal of Antibiotics · 1994 · 31 citations · 6 references
Life SciencesMicrobiologyMolecular BiologyDrug DesignDrug DiscoveryEnzymologyAntibiotic FermentationAntibiotic ProductionEnzyme InhibitionBiological Activity FeaturesFermentation InhibitorsSubstituent Effects On Biological Activity
Streptomyces filipinensis NR 0484 produced a new DNA gyrase inhibitor, cyclothialidine. It showed potent activity against DNA gyrases from Escherichia coli and Micrococcus luteus.
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