Comparison ofR-, S-, andRS-albuterol interaction with human β1 and β2-adrenergic receptors

THE ATTRACTIONS OF PROTEINS FOR SMALL MOLECULES AND IONS

George Scatchard · Annals of the New York Academy of Sciences · 1949 · 19.9K citations

Natural Sciences, Biophysics, Chemistry +9

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

Life Sciences, Biochemistry, Chemical Kinetics +14

cDNA for the human beta 2-adrenergic receptor: a protein with multiple membrane-spanning domains and encoded by a gene whose chromosomal location is shared with that of the receptor for platelet-derived growth factor.

Brian K. Kobilka, Richard A. F. Dixon, Thomas Frielle et al. · Proceedings of the National Academy of Sciences · 1987 · 683 citations · Full text

Life Sciences, Genetics, Molecular Biology +11

Cloning of the cDNA for the human beta 1-adrenergic receptor.

Thomas Frielle, Sheila Collins, Kiefer W. Daniel et al. · Proceedings of the National Academy of Sciences · 1987 · 580 citations · Full text

Life Sciences, Genetics, Molecular Biology +11

Human cardiac beta-adrenergic receptors: Subtype heterogeneity delineated by direct radioligand binding

Gary L. Stiles, Sabrina R. Taylor, Robert J. Lefkowitz · Life Sciences · 1983 · 177 citations

Medicine, Cardiology, Pharmacology +15