Concepedia

Novel human histamine H3 receptor antagonists

Chandra Shah, Laura C. McAtee, J. Guy Breitenbucher, Dale A. Rudolph, Xiaobing Li, Timothy W. Lovenberg, Curt Mazur, Sandy J. Wilson, Nicholas I. Carruthers

Bioorganic & Medicinal Chemistry Letters · 2002 · 40 citations · 19 references

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References

19

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

, , +14

Definition and Antagonism of Histamine H2-receptors

J. W. Black, W. A. M. Duncan, C. J. DURANT et al. · Nature · 1972 · 2.3K citations

, , +12

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

Jean‐Michel Arrang, M. Garbarg, Jean‐Charles Schwartz · Nature · 1983 · 1.6K citations

, , +14

The physiological action of β‐iminazolylethylamine

H. H. Dale, P. P. Laidlaw · The Journal of Physiology · 1910 · 880 citations · Full text

, , +9

Cloning and Functional Expression of the Human Histamine H<sub>3</sub>Receptor

Timothy W. Lovenberg, Barbara Roland, Sandy J. Wilson et al. · Molecular Pharmacology · 1999 · 700 citations · Full text

, , +16