Concepedia

Design and synthesis of a novel peptidomimetic inhibitor of HIV-1 Tat–TAR interactions: Squaryldiamide as a new potential bioisostere of unsubstituted guanidine

Chi‐Wan Lee, Hong Cao, Kozi Ichiyama, Tariq M. Rana

Bioorganic & Medicinal Chemistry Letters · 2005 · 34 citations · 14 references

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14

Tat trans-activates the human immunodeficiency virus through a nascent RNA target

Ben Berkhout, Robert H. Silverman, Kuan‐Teh Jeang · Cell · 1989 · 645 citations

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Oligocarbamate Molecular Transporters:  Design, Synthesis, and Biological Evaluation of a New Class of Transporters for Drug Delivery

Paul A. Wender, Jonathan B. Rothbard, Theodore C. Jessop et al. · Journal of the American Chemical Society · 2002 · 165 citations

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A duodenally absorbable CXC chemokine receptor 4 antagonist, KRH-1636, exhibits a potent and selective anti-HIV-1 activity

Kozi Ichiyama, Sei Yokoyama-Kumakura, Yuetsu Tanaka et al. · Proceedings of the National Academy of Sciences · 2003 · 156 citations

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A facile synthesis of chiral N-protected β-amino alcohols.

Marc Rodriguez, Muriel Llinares, Sylvie Doulut et al. · Tetrahedron Letters · 1991 · 141 citations

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Structure-Based Computational Database Screening, In Vitro Assay, and NMR Assessment of Compounds that Target TAR RNA

Kenneth Lind, Zhihua Du, Koh Fujinaga et al. · Chemistry & Biology · 2002 · 135 citations · Full text

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